SCHEMBL7993940

SCHEMBL7993940

c1cnc2c(-c3cncc(-c4ccsc4)c3)cn(CCN3CCCCC3)c2c1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.74
FLT1 P17948 5/20 0.66
FLT4 P35916 5/20 0.66
CYP2A6 P11509 3/20 0.40
MAPK14 Q16539 2/20 0.39
HTR7 P34969 1/20 0.39
MAOB P27338 1/20 0.36
GSK3B P49841 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990489 0.94 KDR (0.75) KDRFLT1FLT4CYP2A6MAPK14
SCHEMBL7990540 0.91 KDR (0.75) KDRFLT1FLT4CYP2A6MAPK14
SCHEMBL7548593 0.87 KDR (0.57) KDRFLT1FLT4MAPK14GSK3B
SCHEMBL7549006 0.87 KDR (0.75) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7557708 0.87 KDR (0.56) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7549908 0.85 KDR (1.00) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7556531 0.85 KDR (1.00) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7555532 0.84 KDR (0.52) KDRFLT1FLT4MAPK14GSK3B
SCHEMBL7988086 0.83 KDR (0.51) KDRFLT1FLT4MAPK14DRD2
SCHEMBL7551698 0.82 KDR (0.73) KDRFLT1FLT4CYP2A6HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed