SCHEMBL7549928

SCHEMBL7549928

CN1CCNCc2cc(N=C(N)c3cccs3)ccc21

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 13/20 0.65
NOS1 P29475 18/20 0.58
NOS2 P35228 14/20 0.58
CHRM2 P08172 1/20 0.58
ADRA2A P08913 1/20 0.58
CYP2D6 P10635 1/20 0.58
CHRM1 P11229 1/20 0.58
ADRA2B P18089 1/20 0.58
ADRA2C P18825 1/20 0.58
CHRM3 P20309 1/20 0.58
ADRA1D P25100 1/20 0.58
HTR1B P28222 1/20 0.58
ADRA1A P35348 1/20 0.58
ADRA1B P35368 1/20 0.58
KCNH2 Q12809 1/20 0.58
CYP2C19 P33261 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7552153 0.99 NOS3 (0.64) NOS3NOS1NOS2CHRM2ADRA2A
SCHEMBL8177597 0.79 NOS3 (0.91) NOS3NOS1NOS2CHRM2ADRA2A
SCHEMBL7832808 0.79 NOS3 (1.00) NOS3NOS1NOS2CHRM2ADRA2A
SCHEMBL6602318 0.78 NOS1 (0.58) NOS3NOS1NOS2CHRM2ADRA2A
SCHEMBL6602315 0.78 NOS1 (0.58) NOS3NOS1NOS2CHRM2ADRA2A
Hydrochloric Acid SCHEMBL5385353 0.77 NOS1 (0.58) NOS3NOS1NOS2CHRM2ADRA2A
Hydrochloric Acid SCHEMBL5385359 0.77 NOS1 (0.58) NOS3NOS1NOS2CHRM2ADRA2A
SCHEMBL7482742 0.76 NOS3 (0.68) NOS3NOS1NOS2CHRM2ADRA2A
SCHEMBL7550700 0.76 NOS1 (0.49) NOS3NOS1NOS2CHRM2ADRA2A
Hydrochloric Acid SCHEMBL7556788 0.75 NOS1 (0.50) NOS3NOS1NOS2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed