SCHEMBL7549986

SCHEMBL7549986

CC[C@H](NC(=O)OC(C)(C)C)OS(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.44
CTSS P25774 5/20 0.44
CA2 P00918 3/20 0.44
CA1 P00915 2/20 0.44
CA7 P43166 2/20 0.44
CA12 O43570 3/20 0.41
CA14 Q9ULX7 3/20 0.41
SYK P43405 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22196466 1.00 CTSK (0.44) CTSKCTSSCA2CA1CA7
SCHEMBL7831409 1.00 CTSK (0.44) CTSKCTSSCA2CA1CA7
SCHEMBL691120 0.89 CTSK (0.46) CTSKCTSSCA2CA1CA7
SCHEMBL12487322 0.83 CA1 (0.39) CTSKCTSSCA2CA1CA7
SCHEMBL7804172 0.81 KDM4E (0.38) CTSKCTSSCA2CA1CA7
SCHEMBL2341219 0.79 CA1 (0.46) CTSKCTSSCA2CA1CA7
SCHEMBL10650736 0.79 CTSK (0.46) CTSKCTSSCA2CA1CA7
SCHEMBL5146358 0.79 CTSS (0.45) CTSKCTSSCA2CA1CA7
SCHEMBL9527678 0.78 ATM (0.55) CTSKCTSSCA1CA7CA12
SCHEMBL10377816 0.78 ATM (0.55) CTSKCTSSCA1CA7CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202964-A1 CONDENSED INDOLINE DERIVATIVES AND THEIR USE AS 5HT, IN PARTICULAR 5HT2C, RECEPTOR LIGANDS VERNALIS RESEARCH LIMITED (GB) 2002-05-08 EP disclosed
WO-2001012602-A1 CONDENSED INDOLINE DERIVATIVES AND THEIR USE AS 5HT, IN PARTICULAR 5HT2C, RECEPTOR LIGANDS VERNALIS RESEARCH LIMITED (GB) 2001-02-22 WO disclosed