SCHEMBL7551280

SCHEMBL7551280

CC(C)C[C@H](NC(=O)c1ccc(-n2ccnc2)cc1)C(=O)N(C)C#N

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.52
CTSB P07858 7/20 0.51
GFER P55789 2/20 0.49
KMT2A Q03164 1/20 0.49
CTSL P07711 4/20 0.46
CTSS P25774 3/20 0.46
CTSK P43235 3/20 0.46
HTT P42858 1/20 0.45
CYP3A4 P08684 1/20 0.44
BAZ2B Q9UIF8 1/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
F10 P00742 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7554214 0.86 CTSB (0.57) CTSBCTSLCTSSCTSK
SCHEMBL6183202 0.83 CTSL (0.64) TDP1CTSBGFERKMT2ACTSL
SCHEMBL7554406 0.83 CTSB (0.61) CTSBCTSLCTSSCTSK
SCHEMBL7490182 0.82 CTSB (0.52) CTSBCTSLCTSSCTSK
SCHEMBL6182114 0.79 CTSB (0.58) CTSBCTSLCTSSCTSK
SCHEMBL6182791 0.78 CTSB (0.61) CTSBCTSLCTSSCTSK
SCHEMBL6183809 0.78 CTSB (0.61) CTSBCTSLCTSSCTSK
SCHEMBL6183805 0.78 CTSB (0.61) CTSBCTSLCTSSCTSK
SCHEMBL6182874 0.78 CTSB (0.61) CTSBCTSLCTSSCTSK
SCHEMBL7452244 0.78 CTSB (0.61) CTSBKMT2ACTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed