SCHEMBL7553204

SCHEMBL7553204

CCC(N)COCc1cccc(N)c1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.50
MAOB P27338 3/20 0.41
MAOA P21397 2/20 0.41
CYP19A1 P11511 1/20 0.40
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7600364 0.85 TACR1 (0.46) TACR1MAOBMAOACYP19A1
SCHEMBL9507193 0.84 MAOB (0.41) TACR1MAOBMAOACYP19A1TP53
SCHEMBL9066577 0.81 TACR1 (0.57) TACR1
SCHEMBL3621494 0.81 TACR1 (0.57) TACR1
SCHEMBL4088856 0.81 TACR1 (0.57) TACR1
SCHEMBL8011823 0.79 CYP3A4 (0.50) MAOBMAOACYP19A1TP53CYP3A4
SCHEMBL6252491 0.79 ADRB2 (0.44) TACR1MAOBMAOACYP19A1
SCHEMBL6255049 0.79 ADRB2 (0.44) TACR1MAOBMAOACYP19A1
SCHEMBL366865 0.78 MAOB (0.56) MAOBMAOACYP19A1TP53CYP3A4
SCHEMBL2171476 0.78 MAOA (0.47) MAOBMAOACYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214288-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE Targacept Inc. (US) 2002-06-19 EP disclosed
WO-2001017943-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE TARGACEPT, INC. (US) 2001-03-15 WO disclosed
EP-1042274-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-10-11 EP disclosed
WO-2000023418-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-04-27 WO disclosed