SCHEMBL7553508

SCHEMBL7553508

Clc1cccc(-c2cncc(-c3cn(CCN4CCCCC4)c4ccccc34)c2)c1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.69
FLT1 P17948 4/20 0.61
FLT4 P35916 4/20 0.61
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
FLT3 P36888 1/20 0.43
SMYD2 Q9NRG4 1/20 0.41
DRD2 P14416 1/20 0.40
CNR1 P21554 2/20 0.40
CNR2 P34972 2/20 0.40
HTR6 P50406 1/20 0.40
ACP1 P24666 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7556397 0.94 KDR (0.70) KDRFLT1FLT4SMYD2DRD2
SCHEMBL7555476 0.92 KDR (0.58) KDRFLT1FLT4GRIN1GRIN2B
SCHEMBL7551512 0.92 KDR (0.58) KDRFLT1FLT4GRIN1GRIN2B
SCHEMBL7987083 0.91 KDR (0.69) KDRFLT1FLT4CNR1CNR2
SCHEMBL7551441 0.90 KDR (0.71) KDRFLT1FLT4FLT3SMYD2
SCHEMBL7550153 0.89 KDR (0.77) KDRFLT1FLT4FLT3SMYD2
SCHEMBL7548475 0.87 KDR (0.52) KDRFLT1FLT4GRIN1GRIN2B
SCHEMBL7555564 0.87 KDR (0.62) KDRFLT1FLT4GRIN1GRIN2B
SCHEMBL7555743 0.87 KDR (0.62) KDRFLT1FLT4GRIN1GRIN2B
SCHEMBL7550391 0.86 KDR (0.59) KDRFLT1FLT4GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP claimed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP claimed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO claimed
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed