SCHEMBL755513

SCHEMBL755513

C=C(C)C(=O)OCC(C[Si](O[Si](C)(C)C)(O[Si](C)(C)C)O[Si](C)(C)C)OCCCO

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.40
THRB P10828 1/20 0.32
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.30
APEX1 P27695 1/20 0.30
HTT P42858 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL755619 0.90 TSHR (0.40) TSHRTHRBALDH1A1POLBAPEX1
SCHEMBL17983994 0.81 TSHR (0.46) TSHRTHRBALDH1A1
SCHEMBL759922 0.81 TSHR (0.36) TSHRTHRB
SCHEMBL755621 0.79 TSHR (0.37) TSHRTHRB
SCHEMBL3627742 0.75 TSHR (0.49) TSHRTHRBALDH1A1
SCHEMBL9301563 0.75 TSHR (0.53) TSHRTHRBALDH1A1
SCHEMBL3679697 0.74 TSHR (0.40) TSHRTHRB
SCHEMBL663825 0.73 TSHR (0.36) TSHRTHRB
SCHEMBL27823865 0.73 TSHR (0.50) TSHRTHRBALDH1A1POLBAPEX1
SCHEMBL11075198 0.71 TSHR (0.45) TSHRTHRBALDH1A1POLBAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2207825-B8 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE (US) 2012-03-21 EP claimed
EP-2207825-B1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE (US) 2011-06-29 EP claimed
JP-2011502198-A 2011-01-20 JP claimed
EP-2207825-A1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS Johnson & Johnson Vision Care, Inc. (US) 2010-07-21 EP claimed
EP-1809344-B1 BIOMEDICAL DEVICES CONTAINING AMPHIPHILIC BLOCK COPOLYMERS JOHNSON & JOHNSON VISION CARE (US) 2010-01-20 EP claimed
WO-2009058207-A1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE, INC. (US) 2009-05-07 WO claimed
US-20090111905-A1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE, INC. 2009-04-30 US claimed
EP-2207825-B8 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE (US) 2012-03-21 EP disclosed
EP-2207825-B1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE (US) 2011-06-29 EP disclosed
EP-2207825-A1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS Johnson & Johnson Vision Care, Inc. (US) 2010-07-21 EP disclosed
WO-2009058207-A1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE, INC. (US) 2009-05-07 WO disclosed
US-20090111905-A1 PROCESS FOR FORMING RANDOM (METH)ACRYLATE CONTAINING PREPOLYMERS JOHNSON & JOHNSON VISION CARE, INC. 2009-04-30 US disclosed