SCHEMBL7556147

SCHEMBL7556147

O=C(NC[C]1CCCCCCC1)c1ccc(OC2CCNCC2)cc1Cl.[CH2].[CH2]

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.52
HRH3 Q9Y5N1 3/20 0.46
UTS2R Q9UKP6 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ROCK1 Q13464 2/20 0.38
KDM1A O60341 2/20 0.38
HRH1 P35367 3/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CCR3 P51677 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5398913 0.92 P2RX7 (0.63) P2RX7HRH3UTS2RALDH1A1SMN1; SMN2
SCHEMBL7555599 0.83 HRH3 (0.42) P2RX7HRH3NPC1RAB9APOLB
SCHEMBL7515669 0.79 P2RX7 (0.48) P2RX7HRH3SMN1; SMN2HRH1CCR3
SCHEMBL7556141 0.77 P2RX7 (0.85) P2RX7
SCHEMBL7554565 0.76 P2RX7 (0.51) P2RX7NPC1RAB9APOLBHPGD
SCHEMBL7518675 0.75 ESRRB (0.49) P2RX7NPC1RAB9APOLBHPGD
SCHEMBL7555457 0.75 P2RX7 (0.47) P2RX7
SCHEMBL7559238 0.74 HPGD (0.46) P2RX7NPC1RAB9APOLBHPGD
SCHEMBL7603269 0.73 P2RX7 (0.45) P2RX7HPGDALDH1A1SMN1; SMN2
SCHEMBL21434774 0.72 KDM4E (0.55) P2RX7HRH3NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492355-B1 Adamantane derivatives ASTRAZENECA AB (SE) 2002-12-10 US disclosed
EP-1171432-A1 ADAMANTANE DERIVATIVES AstraZeneca AB (SE) 2002-01-16 EP disclosed
WO-2000061569-A1 ADAMANTANE DERIVATIVES ASTRAZENECA AB (SE) 2000-10-19 WO disclosed