SCHEMBL7558696

SCHEMBL7558696

CN1C(=O)CCN(C(=O)c2ccccc2)[C@H]1C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ACHE P22303 1/20 0.40
POLB P06746 1/20 0.39
ADRB2 P07550 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PIK3CD O00329 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
RBP4 P02753 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7558692 1.00 PARP1 (0.42) PARP1ALDH1A1TSHRRECQLSMN1; SMN2
SCHEMBL8232622 1.00 PARP1 (0.42) PARP1ALDH1A1TSHRRECQLSMN1; SMN2
SCHEMBL8238415 0.86 RBP4 (0.42) ALDH1A1TSHRRECQLSMN1; SMN2ACHE
SCHEMBL9706890 0.86 RBP4 (0.42) ALDH1A1TSHRRECQLSMN1; SMN2ACHE
SCHEMBL7193232 0.86 RBP4 (0.42) ALDH1A1TSHRRECQLSMN1; SMN2ACHE
SCHEMBL22541399 0.82 GAA (0.41) ALDH1A1SMN1; SMN2POLBMAPTL3MBTL1
SCHEMBL1704378 0.75 CNR2 (0.36) ALDH1A1
SCHEMBL3054057 0.75 CNR2 (0.36) ALDH1A1
SCHEMBL8259156 0.74 TSHR (0.41) PARP1ALDH1A1TSHRRECQLSMN1; SMN2
SCHEMBL8257096 0.74 TSHR (0.41) PARP1ALDH1A1TSHRRECQLSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002066417-A1 METHOD FOR THE PRODUCTION OF THE ENANTIOMERS OF 2-SUBSTITUTED BETA AMINO ACIDS CHIROBLOCK GMBH (DE) 2002-08-29 WO disclosed
US-6372936-B1 REACTING AMINO PROTECTED RACEMIC 3-AMINO-2-METHYL PROPIONIC ACID WITH ENANTIOMER OF CHIRAL AMINE TO FORM DIASTEREOMERIC SALTS, RECRYSTALLIZING SALTS FROM ETHYL ACETATE TO SEPARATE, RELEASING RESOLVED ACID WITH SOLUTION OF INORGANIC BASE ELI LILLY AND COMPANY 2002-04-16 US disclosed
EP-1059286-A1 Optical resolution of aminoisobutyric acid ELI LILLY AND COMPANY (US) 2000-12-13 EP disclosed