SCHEMBL8259156

SCHEMBL8259156

CCC(C)[C@H]1N(C)C(=O)CCN1C(=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 2/20 0.41
ABCB1 P08183 3/20 0.41
ABCG2 Q9UNQ0 2/20 0.41
PIK3CD O00329 1/20 0.40
PARP1 P09874 1/20 0.39
BLM P54132 1/20 0.39
MTNR1B P49286 1/20 0.38
RECQL P46063 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8257096 1.00 TSHR (0.41) TSHRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7558696 0.74 PARP1 (0.42) TSHRL3MBTL1ALDH1A1ABCB1ABCG2
SCHEMBL7558692 0.74 PARP1 (0.42) TSHRL3MBTL1ALDH1A1ABCB1ABCG2
SCHEMBL8232622 0.74 PARP1 (0.42) TSHRL3MBTL1ALDH1A1ABCB1ABCG2
SCHEMBL19386648 0.66 ALDH1A1 (0.44) ALDH1A1PIK3CDBLMHPGD
SCHEMBL9197399 0.65 ABCB1 (0.41) TSHRL3MBTL1ABCB1ABCG2PARP1
SCHEMBL9220425 0.65 L3MBTL1 (0.45) TSHRL3MBTL1ALDH1A1ABCB1ABCG2
SCHEMBL8028682 0.64 ACHE (0.44) TSHRALDH1A1ABCB1PIK3CDRECQL
SCHEMBL7338840 0.63 ALDH1A1 (0.61) CYP2D6CYP2C9CYP2C19ALDH1A1BLM
SCHEMBL9873550 0.63 ALDH1A1 (0.45) L3MBTL1ALDH1A1PIK3CDBLMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006120544-A1 β-AMINO ACID DERIVATIVES PFIZER LIMITED (GB) 2006-11-16 WO disclosed