SCHEMBL7559455

SCHEMBL7559455

CC(C)(C)OC(=O)NC1(C(=O)NC(CCc2ccccc2)C(O)c2nc3ccccc3o2)CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.40
CTSS P25774 3/20 0.37
CTSK P43235 1/20 0.37
CTSB P07858 2/20 0.36
CTSL P07711 1/20 0.36
FAAH O00519 3/20 0.36
CXCR2 P25025 1/20 0.36
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
MAPT P10636 3/20 0.35
ATM Q13315 1/20 0.35
PTPN2 P17706 2/20 0.34
PTPN1 P18031 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 2/20 0.34
TSHR P16473 2/20 0.34
HSD17B10 Q99714 2/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5731226 0.86 CTSK (0.46) CTSSCTSKMAPTATMALDH1A1
SCHEMBL5731227 0.86 CTSK (0.46) CTSSCTSKMAPTATMALDH1A1
SCHEMBL6347225 0.77 KLK5 (0.49) CTSSCTSKCTSBCTSLMAPT
SCHEMBL6415412 0.76 NPC1 (0.35) CTSKMAPTPTPN2PTPN1TP53
SCHEMBL5736602 0.76 NPC1 (0.42) CTSSCTSKCTSLMAPTATM
SCHEMBL5736600 0.76 NPC1 (0.42) CTSSCTSKCTSLMAPTATM
SCHEMBL6062065 0.75 CTSS (0.41) CTSSCTSKMAPTATMRAB9A
SCHEMBL6062057 0.75 CTSS (0.41) CTSSCTSKMAPTATMRAB9A
SCHEMBL6062062 0.75 CTSS (0.41) CTSSCTSKMAPTATMRAB9A
SCHEMBL6696297 0.75 CTSS (0.41) CTSSCTSKMAPTATMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002023784-A2 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-03-21 WO disclosed