SCHEMBL7560541

SCHEMBL7560541

CCOC(=O)c1ccc(S(=O)(=O)N(C)c2ccc(OC[C@@H](O)CNC(C)(C)Cc3ccc4ccccc4c3)c(C#N)c2)cc1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASR P41180 18/20 0.65
CYP2D6 P10635 9/20 0.65
SLC6A2 P23975 8/20 0.65
SLC6A4 P31645 8/20 0.65
SLC6A3 Q01959 8/20 0.65
KCNH2 Q12809 8/20 0.65
ADRB2 P07550 5/20 0.65
ADRB3 P13945 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7560544 1.00 CASR (0.65) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7560533 1.00 CASR (0.65) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7560527 0.86 CASR (0.69) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7563669 0.84 CASR (0.48) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7607141 0.84 CASR (0.71) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6863014 0.82 CASR (0.62) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6863019 0.82 CASR (0.62) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7606278 0.82 CASR (0.70) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7606286 0.82 CASR (0.70) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6862107 0.82 CASR (0.61) CASRCYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002072760-A2 PCRA HELICASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-09-19 WO claimed
WO-2002072760-A2 PCRA HELICASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-09-19 WO disclosed