SCHEMBL7563669

SCHEMBL7563669

CCOC(=O)c1ccc(S(=O)(=O)N(C)c2ccc(OC[C@H](O)C[N+](C)(C)CCc3ccc4ccccc4c3)c(C#N)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASR P41180 6/20 0.48
SLC6A2 P23975 4/20 0.48
SLC6A4 P31645 4/20 0.48
SLC6A3 Q01959 4/20 0.48
KCNH2 Q12809 4/20 0.48
CYP2D6 P10635 4/20 0.48
ADRB2 P07550 2/20 0.48
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
POLB P06746 3/20 0.36
ALDH1A1 P00352 2/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
KEAP1 Q14145 2/20 0.34
NFE2L2 Q16236 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7560533 0.84 CASR (0.65) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7560544 0.84 CASR (0.65) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7560541 0.84 CASR (0.65) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8169408 0.81 KEAP1 (0.45) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8167993 0.81 ALDH1A1 (0.47) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6220841 0.78 CASR (0.63) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8172490 0.78 CASR (0.46) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7563830 0.78 CASR (0.46) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8172146 0.77 CASR (0.49) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8166977 0.75 KCNH2 (0.49) CASRSLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002072760-A2 PCRA HELICASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-09-19 WO claimed