SCHEMBL7562425

SCHEMBL7562425

Cc1c(Br)cc2c(c1C(C)C)OCC2(C)C

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 6/20 0.32
PTGS2 P35354 6/20 0.32
ALOX5 P09917 4/20 0.32
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7568295 0.77 PTGS2 (0.41) PTGS1PTGS2ALOX5
SCHEMBL25181143 0.74 PTGS2 (0.36) PTGS1PTGS2ALOX5NOTUM
SCHEMBL7564517 0.72 PTGS2 (0.41) PTGS1PTGS2ALOX5
SCHEMBL7563291 0.72 PTGS2 (0.38) PTGS1PTGS2ALOX5
SCHEMBL2489432 0.72 AHR (0.38) PTGS1PTGS2ALOX5NOTUM
SCHEMBL6756512 0.70 GABRA1 (0.41) PTGS1PTGS2ALOX5NOTUM
SCHEMBL5659858 0.70 PTGS2 (0.36) PTGS1PTGS2ALOX5
SCHEMBL7564521 0.70 PTGS2 (0.34) PTGS1PTGS2ALOX5NOTUM
SCHEMBL7564258 0.69 AKR1C3 (0.38)
SCHEMBL3478661 0.69 PTGS2 (0.34) PTGS1PTGS2ALOX5NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228055-A1 DIHYDROAMINOBENZO[B]- AND [C]FURANS AS RETINOID-LIKE AGENTS Allergan Sales, Inc. (US) 2002-08-07 EP disclosed
WO-2001012618-A1 DIHYDROAMINOBENZO[B]- AND [C]FURANS AS RETINOID-LIKE AGENTS ALLERGAN SALES, INC. (US) 2001-02-22 WO disclosed
US-6093838-A FOR TREATING SKIN-RELATED DISEASES, INCLUDING ACTINIC KERATOSES, ARSENIC KERATOSES, ECZEMA ALLERGAN SALES, INC. (US) 2000-07-25 US disclosed