SCHEMBL7562774

SCHEMBL7562774

CC(C)c1[c]c(-c2ccc(F)cc2)nc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.43
TNKS O95271 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
GRM2 Q14416 1/20 0.41
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 1/20 0.39
CYP19A1 P11511 1/20 0.39
SCN9A Q15858 4/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM1A O60341 1/20 0.38
CCNE2 O96020 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302519 0.73 ADORA2A (0.43) ADORA2ATNKSTNKS2PARP2GRM2
SCHEMBL8321756 0.70 GCGR (0.46) ADORA2ATNKSTNKS2PARP2GRM2
SCHEMBL10345401 0.69 CYP19A1 (0.56) ADORA2AALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL14544897 0.68 GCGR (0.44) ADORA2ATNKSTNKS2PARP2ALDH1A1
SCHEMBL8877398 0.67 HMGCR (0.51) ADORA2ATNKSTNKS2PARP2GRM2
SCHEMBL22876085 0.67 GCGR (0.58) ADORA2A
SCHEMBL577952 0.66 MAPK14 (0.47) ADORA2ATNKSTNKS2PARP2GRM2
SCHEMBL12525154 0.66 ALDH1A1 (0.61) ADORA2AGRM2ALDH1A1SMN1; SMN2KMT2A
SCHEMBL8877962 0.66 HMGCR (0.53) ADORA2AALDH1A1SMN1; SMN2SCN9AMAPT
Methane SCHEMBL10345343 0.66 HMGCR (0.50) ADORA2ASCN9AMAPK10MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705837-B1 Preparation of 3-Oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES (JP) 2002-08-07 EP disclosed
US-5744604-A Preparation of 3-oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1998-04-28 US disclosed
US-5677455-A Preparation of 3-oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0705837-A2 Preparation of 3-Oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1996-04-10 EP disclosed