SCHEMBL7562782

SCHEMBL7562782

O=C1c2c(Br)c(Br)c(Br)c(Br)c2C(=O)N1CO

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 7/20 0.41
CA2 P00918 6/20 0.41
CA7 P43166 6/20 0.41
CA1 P00915 5/20 0.41
CA12 O43570 5/20 0.41
CA4 P22748 2/20 0.39
TSHR P16473 1/20 0.35
HIPK2 Q9H2X6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912698 0.81 CA9 (0.44) CA9CA2CA7CA1CA12
SCHEMBL29366486 0.79 CA9 (0.49) CA9CA2CA7CA1CA12
SCHEMBL94242 0.79 CA9 (0.49) CA9CA2CA7CA1CA12
SCHEMBL6046957 0.79 CA9 (0.43) CA9CA2CA7CA1CA12
SCHEMBL10999370 0.77 CA9 (0.42) CA9CA2CA7CA1CA12
SCHEMBL11295187 0.75 CA1 (0.46) CA9CA2CA7CA1CA12
SCHEMBL3692053 0.75 F2 (0.43) CA9CA2CA7CA1CA12
SCHEMBL5090368 0.75 CA12 (0.46) CA9CA2CA7CA1CA12
SCHEMBL10570526 0.73 CA12 (0.45) CA9CA2CA7CA1CA12
SCHEMBL6570337 0.73 CA12 (0.45) CA9CA2CA7CA1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1376182-A Process for improving the toughness of PCT formulations by adding rubber impact modifiers EASTMAN CHEM CO (US) 2002-10-23 CN disclosed
CN-1374980-A Improved PCT formulations containing halogenated imides, sodium antimonate and reinforcing fibers EASTMAN CHEM CO (US) 2002-10-16 CN disclosed
EP-1228130-A2 IMPROVED PCT FORMULATIONS CONTAINING HALOGENATED IMIDES, SODIUM ANTIMONATE, AND REINFORCING FIBERS EASTMAN CHEMICAL COMPANY (US) 2002-08-07 EP disclosed
EP-1214376-A1 PROCESS FOR IMPROVING THE TOUGHNESS OF PCT FORMULATIONS BY ADDING RUBBER IMPACT MODIFIERS EASTMAN CHEMICAL COMPANY (US) 2002-06-19 EP disclosed
US-6277905-B1 BLENDING POLYCYCLOHEXYLENEDIMETHYLENE TEREPHTHALATE, RUBBER IMPACT MODIFIER, HALOGENATED ORGANIC COMPOUND CONTAINING AT LEAST ONE IMIDE GROUP AND HAVING SPECIFIED MELTING POINT, REINFORCING FIBER AND SELECTED PHOSPHITE EASTMAN CHEMICAL COMPANY 2001-08-21 US disclosed
WO-2001027200-A2 REINFORCED PCT FORMULATIONS CONTAINING HALOGENATED IMIDES AND IMPACT MODIFIERS EASTMAN CHEMICAL COMPANY (US) 2001-04-19 WO disclosed
WO-2001025325-A2 IMPROVED PCT FORMULATIONS CONTAINING HALOGENATED IMIDES, SODIUM ANTIMONATE, AND REINFORCING FIBERS EASTMAN CHEMICAL COMPANY (US) 2001-04-12 WO disclosed
WO-2001021701-A1 IMPROVED POLYESTER FORMULATIONS CONTAINING HALOGENATED IMIDE(S), PENTAERYTHRITOL ESTER(S) AND REINFORCING FIBER EASTMAN CHEMICAL COMPANY (US) 2001-03-29 WO disclosed
WO-2001021700-A1 PROCESS FOR IMPROVING THE MELT STABILITY OF HALOGENATED IMIDES IN PCT FORMULATIONS BY ADDITION OF SODIUM ANTIMONATE EASTMAN CHEMICAL COMPANY (US) 2001-03-29 WO disclosed
WO-2001021704-A1 PROCESS FOR IMPROVING THE OVEN AGING STABILITY OF PCT FORMULATIONS BY ADDITION OF PHENOXY COMPOUND(S) EASTMAN CHEMICAL COMPANY (US) 2001-03-29 WO disclosed
WO-2001021703-A1 PROCESS FOR IMPROVING FLAMMABILITY CHARACTERISTICS OF POLYESTER FORMULATIONS BY ADDING PENTAERYTHRITOL ESTER(S) EASTMAN CHEMICAL COMPANY (US) 2001-03-29 WO disclosed
WO-2001021710-A1 PROCESS FOR IMPROVING THE TOUGHNESS OF PCT FORMULATIONS BY ADDING RUBBER IMPACT MODIFIERS EASTMAN CHEMICAL COMPANY (US) 2001-03-29 WO disclosed
WO-2001021702-A1 IMPROVED PCT FORMULATIONS CONTAINING HALOGENATED IMIDES, PHENOXY COMPOUND(S) AND REINFORCING FIBERS EASTMAN CHEMICAL COMPANY (US) 2001-03-29 WO disclosed
EP-0146104-A2 Polyester thermoplastic molding compositions with good mold release MOBAY CORPORATION (US) 1985-06-26 EP disclosed
EP-0029930-B1 USE OF POLYETHYLENE TEREPHTHALATE MOULDING MASSES CONTAINING AN ORGANIC IMIDE IN THE PREPARATION OF CRYSTALLINE MOULDINGS BY INJECTION MOULDING AT LOW MOULD TEMPERATURES BAYER AG (DE) 1984-02-15 EP disclosed
EP-0083796-A1 Flame-resistant moulding masses based on polyethylene terephthalate, process for its preparation and its use in the production of articles BAYER AG (DE) 1983-07-20 EP disclosed
EP-0030618-A1 Flame-resistant moulding masses based on polyethyleneterephthalate, process for their preparation and their use in producing mouldings BAYER AG (DE) 1981-06-24 EP disclosed
EP-0029930-A1 Use of polyethylene terephthalate moulding masses containing an organic imide in the preparation of crystalline mouldings by injection moulding at low mould temperatures BAYER AG (DE) 1981-06-10 EP disclosed
US-4254011-A CONTAINING A TWO-PHASE CROSSLINKED POLYACRYLATE BAYER AKTIENGESELLSCHAFT (DE) 1981-03-03 US disclosed
US-4003862-A N-substituted tetrahalophthalimides as flame retardants MICHIGAN CHEMICAL CORPORATION (US) 1977-01-18 US disclosed