SCHEMBL7563232

SCHEMBL7563232

C=CCOC(=O)c1cccc(N)c1C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.72
HSD17B10 Q99714 7/20 0.72
TSHR P16473 3/20 0.72
CYP3A4 P08684 2/20 0.63
MAPT P10636 3/20 0.43
POLB P06746 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 3/20 0.43
TP53 P04637 2/20 0.43
HPGD P15428 2/20 0.43
CDC25B P30305 2/20 0.42
MAPK1 P28482 2/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
RAB9A P51151 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11181389 0.89 CYP3A4 (0.73) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL250686 0.86 ALDH1A1 (0.60) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL5339693 0.84 ALDH1A1 (0.77) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL9422015 0.84 CYP3A4 (0.67) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL759012 0.84 ALDH1A1 (1.00) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL8788785 0.83 ALDH1A1 (0.74) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL27597729 0.83 CYP3A4 (0.65) ALDH1A1HSD17B10TSHRCYP3A4MAPT
Hydrochloric Acid SCHEMBL28469611 0.83 ALDH1A1 (0.97) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL5095287 0.82 ALDH1A1 (0.68) ALDH1A1HSD17B10TSHRCYP3A4MAPT
SCHEMBL717606 0.82 ALDH1A1 (0.74) ALDH1A1HSD17B10TSHRCYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178958-A2 N-CYANOMETHYL AMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-02-13 EP disclosed
WO-2000055125-A2 N-CYANOMETHYL AMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed