SCHEMBL7564762

SCHEMBL7564762

O=C(O)c1cccc2c(=O)c3cc(Br)ccc3[nH]c12

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 2/20 0.69
AR P10275 1/20 0.51
CCNB2 O95067 1/20 0.45
CCNE2 O96020 1/20 0.45
CDK1 P06493 1/20 0.45
CDK4 P11802 1/20 0.45
CCNB1 P14635 1/20 0.45
CCND1 P24385 1/20 0.45
CCNE1 P24864 1/20 0.45
CDK2 P24941 1/20 0.45
CCNB3 Q8WWL7 1/20 0.45
RXFP1 Q9HBX9 3/20 0.44
PRNP P04156 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PPARG P37231 1/20 0.44
HIF1A Q16665 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NR2E3 Q9Y5X4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10857797 0.89 PBRM1 (0.69) PBRM1ARCCNB2CCNE2CDK1
SCHEMBL2440948 0.83 PBRM1 (0.69) PBRM1MEN1KMT2AGFERMAPT
SCHEMBL7568234 0.83 PBRM1 (0.69) PBRM1CYP2C19KMT2AGFERMAPT
SCHEMBL7570750 0.82 PBRM1 (0.72) PBRM1MEN1KMT2AGFERMAPT
SCHEMBL4943278 0.82 PBRM1 (1.00) PBRM1CYP1A2CYP2C19MEN1KMT2A
SCHEMBL29801740 0.82 PBRM1 (1.00) PBRM1CYP1A2CYP2C19MEN1KMT2A
SCHEMBL27450150 0.81 PARP1 (0.50) PBRM1ARCCNB2CCNE2CDK1
SCHEMBL8789976 0.80 PBRM1 (0.64) PBRM1MEN1KMT2AGFERMAPT
SCHEMBL7567402 0.80 PBRM1 (0.64) PBRM1KDM4EDHFR
SCHEMBL7565942 0.80 PBRM1 (0.64) PBRM1GFERMAPTTDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1116285-C Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2003-07-30 CN disclosed
EP-0934278-B1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LTD (GB) 2002-09-04 EP disclosed
US-6114332-A BACTERICIDES XENOVA LIMITED (GB) 2000-09-05 US disclosed
CN-1240430-A Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2000-01-05 CN disclosed
EP-0934278-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1999-08-11 EP disclosed
WO-1998017650-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1998-04-30 WO disclosed