SCHEMBL7564902

SCHEMBL7564902

COc1ccc2nc(S(=O)(=O)C(Br)(Br)Br)sc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C19 P33261 2/20 0.54
PDK1 Q15118 1/20 0.52
CA2 P00918 11/20 0.52
CA1 P00915 2/20 0.51
KMT2A Q03164 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CA12 O43570 1/20 0.51
LMNA P02545 1/20 0.51
CA3 P07451 1/20 0.51
PKM P14618 1/20 0.51
CA4 P22748 1/20 0.51
CA6 P23280 1/20 0.51
CA5A P35218 1/20 0.51
CA7 P43166 1/20 0.51
HIF1A Q16665 1/20 0.51
CA9 Q16790 1/20 0.51
CA13 Q8N1Q1 1/20 0.51
TDP1 Q9NUW8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748302 0.84 CYP1A2 (0.58) CYP1A2CYP3A4CYP2C19PDK1CA2
SCHEMBL32679829 0.81 CA2 (0.59) CYP1A2CYP3A4CYP2C19PDK1CA2
SCHEMBL299010 0.75 CYP1A2 (0.67) CYP1A2CYP3A4CYP2C19PDK1KMT2A
SCHEMBL3275548 0.73 PSMB8 (0.66) PDK1CA2CA1KMT2ACA12
SCHEMBL4273826 0.73 CYP1A2 (0.59) CYP1A2CYP3A4CYP2C19PDK1KMT2A
SCHEMBL25492543 0.72 CA2 (0.44) CA2CA1KMT2AKDM4ECA12
SCHEMBL3634489 0.72 HSD17B1 (0.63) CYP1A2CYP3A4CYP2C19PDK1KMT2A
SCHEMBL11823356 0.72 NPC1 (0.52) CA2PKMNPC1RAB9ASMN1; SMN2
SCHEMBL11973204 0.72 DYRK1A (0.46) CA2CA1KDM4ECA12LMNA
SCHEMBL422166 0.72 CYP1A2 (0.67) CYP1A2CYP3A4CYP2C19PDK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0720053-B1 Photosensitive resin composition, photosensitive printing plate and method of manufacturing printing master plate TOKYO OHKA KOGYO CO LTD (JP) 2002-09-04 EP claimed
US-5885746-A COMPRISING A POLYMER BINDER, A MONOMER, A PHOTOINITIATOR ACTIVATED BY VISIBLE LASER LIGHT, A PHOTOSENSITIVE ACID-GENERATING AGENT AND A CHROMOGEN; OFFSET PRINTING; STORAGE STABILITY; RESOLUTION; MATERIALS HANDLING; EFFICIENCY TOKYO OHKA KOGYO CO., LTD. (JP) 1999-03-23 US claimed
EP-0720053-A2 Photosensitive resin composition, photosensitive printing plate and method of manufacturing printing master plate TOKYO OHKA KOGYO CO., LTD. (JP) 1996-07-03 EP claimed
US-4094676-A Non-silver salt type photosensitive composition ASAHI KASEI KOGYO KABUSHIKI KAISHA (JA) 1978-06-13 US claimed
EP-0720053-B1 Photosensitive resin composition, photosensitive printing plate and method of manufacturing printing master plate TOKYO OHKA KOGYO CO LTD (JP) 2002-09-04 EP disclosed
US-5885746-A COMPRISING A POLYMER BINDER, A MONOMER, A PHOTOINITIATOR ACTIVATED BY VISIBLE LASER LIGHT, A PHOTOSENSITIVE ACID-GENERATING AGENT AND A CHROMOGEN; OFFSET PRINTING; STORAGE STABILITY; RESOLUTION; MATERIALS HANDLING; EFFICIENCY TOKYO OHKA KOGYO CO., LTD. (JP) 1999-03-23 US disclosed
EP-0720053-A2 Photosensitive resin composition, photosensitive printing plate and method of manufacturing printing master plate TOKYO OHKA KOGYO CO., LTD. (JP) 1996-07-03 EP disclosed
US-4465761-A HALO COMPOUND, LEUCO DYE, AROMATIC AMINE SENSITIZER, BINDER AND ALIPHATIC AMINE; ANTIFOGGING AGENTS ORIENTAL PHOTO INDUSTRIES CO., LTD. (JP) 1984-08-14 US disclosed
EP-0026859-B1 IMAGE-FORMING PHOTOSENSITIVE COMPOSITION, PHOTOSENSITIVE COATING SOLUTION AND PHOTOSENSITIVE SHEET COMPRISING THIS COMPOSITION ORIENTAL PHOTO INDUSTRIES, CO., LTD. (JP) 1983-10-05 EP disclosed
US-4094676-A Non-silver salt type photosensitive composition ASAHI KASEI KOGYO KABUSHIKI KAISHA (JA) 1978-06-13 US disclosed
US-3957513-A Method of free radical photography utilizing a short light flash for exposure ASAHI KASEI KOGYO KABUSHIKI KAISHA (JA) 1976-05-18 US disclosed