SCHEMBL7565325

SCHEMBL7565325

CC(C)CC(NC(=O)OC(C)(C)C)C(=O)NC1CCCN(S(=O)(=O)c2cccc[n+]2[O-])CC1O

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.45
MAPK1 P28482 1/20 0.39
CACNA1B Q00975 2/20 0.38
CCKAR P32238 1/20 0.37
CTSL P07711 2/20 0.36
CTSS P25774 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687294 1.00 CTSK (0.45) CTSKMAPK1CACNA1BCCKARCTSL
SCHEMBL7207130 0.89 CTSK (0.45) CTSKCACNA1BCTSLCTSSKMT2A
SCHEMBL7036592 0.87 CTSK (0.51) CTSKMAPK1CACNA1BCCKARCTSL
SCHEMBL4902191 0.87 CTSK (0.51) CTSKMAPK1CACNA1BCCKARCTSL
SCHEMBL5099105 0.85 CTSK (0.47) CTSKMAPK1
SCHEMBL5099103 0.85 CTSK (0.47) CTSKMAPK1
SCHEMBL5099268 0.84 CTSK (0.41) CTSKCACNA1BCTSLCTSS
SCHEMBL7426616 0.84 CTSK (0.44) CTSKCACNA1BCTSLCTSSMEN1
SCHEMBL5582054 0.84 CACNA1B (0.47) CTSKCACNA1BKMT2A
SCHEMBL5582055 0.84 CACNA1B (0.47) CTSKCACNA1BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed