SCHEMBL7565531

SCHEMBL7565531

C[C@@H](CC(N)=O)CC(=O)NC1CCCN(CCc2ccccc2)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
XIAP P98170 1/20 0.42
BIRC2 Q13490 1/20 0.42
CTSK P43235 4/20 0.41
CTSL P07711 2/20 0.40
CTSS P25774 2/20 0.40
HRH3 Q9Y5N1 1/20 0.39
DRD3 P35462 1/20 0.38
OPRM1 P35372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7565521 1.00 SIGMAR1 (0.43) SIGMAR1XIAPBIRC2CTSKCTSL
SCHEMBL6771044 0.85 CTSK (0.44) CTSKCTSLCTSS
SCHEMBL6771052 0.85 CTSK (0.44) CTSKCTSLCTSS
SCHEMBL5099108 0.80 CTSK (0.51) SIGMAR1XIAPBIRC2CTSKCTSL
SCHEMBL6599017 0.78 CTSK (0.43) SIGMAR1XIAPBIRC2CTSKCTSL
SCHEMBL4924362 0.73 CTSK (0.56) CTSKCTSLCTSS
SCHEMBL6592566 0.73 CTSK (0.36) CTSKCTSLCTSS
SCHEMBL6766533 0.72 CTSK (0.36) CTSKCTSLCTSS
SCHEMBL6765207 0.72 CYP3A4 (0.45) CTSK
SCHEMBL6761962 0.71 POLB (0.46) CTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed