SCHEMBL7566083

SCHEMBL7566083

COc1ccc(C(C)=O)c(OCCCC(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
POLB P06746 1/20 0.52
PTPN1 P18031 1/20 0.52
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
CYP3A4 P08684 1/20 0.51
MAPK1 P28482 1/20 0.51
HTT P42858 2/20 0.51
FFAR1 O14842 1/20 0.51
FFAR4 Q5NUL3 1/20 0.51
CYSLTR2 Q9NS75 5/20 0.51
CYSLTR1 Q9Y271 5/20 0.51
TSHR P16473 1/20 0.50
LMNA P02545 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21098685 0.90 CYSLTR2 (0.53) MAPTL3MBTL1HTTFFAR1FFAR4
SCHEMBL30991357 0.88 LMNA (0.52) MAPTL3MBTL1POLBALDH1A1HPGD
SCHEMBL9525503 0.84 LMNA (0.54) MAPTL3MBTL1POLBALDH1A1HPGD
SCHEMBL1114933 0.83 POLB (0.64) MAPTL3MBTL1POLBPTPN1ALDH1A1
SCHEMBL2225179 0.83 LMNA (0.57) MAPTL3MBTL1POLBPTPN1ALDH1A1
SCHEMBL28382637 0.82 MAPT (0.54) MAPTL3MBTL1POLBALDH1A1HPGD
SCHEMBL1115022 0.80 LMNA (0.63) MAPTL3MBTL1POLBPTPN1ALDH1A1
SCHEMBL17594055 0.80 POLB (0.50) POLBPTPN1FFAR1FFAR4CYSLTR2
SCHEMBL3182853 0.80 NPC1 (0.68) MAPTL3MBTL1POLBPTPN1ALDH1A1
SCHEMBL7497130 0.80 KDM4E (0.61) MAPTL3MBTL1POLBALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0689845-B1 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID CO (US) 2002-09-04 EP disclosed
US-5877296-A REACTING DISULFIDE ANALOGS OF CALICHEAMICIN FAMILY WITH A CARRIER SUCH AS PROTEIN, PEPTIDE, MONO AND POLYCLONAL ANTIBODIES, THEIR ANTIGEN-RECOGNIZING FRAGMENTS AND CHEMICALLY OR GENETICALLY ENGINEERED COUNTERPARTS AMERICAN CYANAMID COMPANY (US) 1999-03-02 US disclosed
US-5773001-A ANTIGROWTH AGENTS AMERICAN CYANAMID COMPANY (US) 1998-06-30 US disclosed
US-5767285-A USEFUL FOR CONSTRUCTING DRUG CONJUGATES; ANTIBIOTIC ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY (US) 1998-06-16 US disclosed
US-5739116-A DISULFIDE DERIVATIVE OF CALICHEAMICIN FAMILY; ANTITUMOR ANTIBIOTICS AMERICAN CYANAMID COMPANY (US) 1998-04-14 US disclosed
EP-0689845-A2 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID COMPANY (US) 1996-01-03 EP disclosed