SCHEMBL7566830

SCHEMBL7566830

C=CCn1nc(OCC(=O)c2cccs2)c(-c2ccc(F)cc2)c1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.47
PTGS1 P23219 5/20 0.41
CA9 Q16790 1/20 0.35
HPGD P15428 2/20 0.35
CTSB P07858 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7536789 0.90 PTGS2 (0.43) PTGS2PTGS1CA9HPGDCTSB
SCHEMBL6619309 0.90 PTGS2 (0.43) PTGS2PTGS1CA9HPGDCTSB
SCHEMBL7535016 0.81 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL6622652 0.77 PTGS2 (0.41) PTGS2PTGS1HPGDMAPT
SCHEMBL7665809 0.77 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL7671385 0.76 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL7669405 0.76 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL7670248 0.76 PTGS2 (0.45) PTGS2PTGS1MAPTKMT2A
SCHEMBL7670052 0.74 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL6622930 0.73 PTGS2 (0.46) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472416-B1 Sulfonylphenylpyrazole compounds useful as COX-2 inhibitors ABBOTT LABORATORIES 2002-10-29 US disclosed
EP-1206474-A1 SULFONYLPHENYLPYRAZOLE COMPOUNDS USEFUL AS COX-2 INHIBITORS ABBOTT LABORATORIES (US) 2002-05-22 EP disclosed
WO-2001016138-A1 SULFONYLPHENYLPYRAZOLE COMPOUNDS USEFUL AS COX-2 INHIBITORS ABBOTT LABORATORIES (US) 2001-03-08 WO disclosed