SCHEMBL7567690

SCHEMBL7567690

COc1cn(Cc2ccc(OCc3ccccc3)cc2)nc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.51
FAAH O00519 1/20 0.49
MGLL Q99685 1/20 0.49
KMT2A Q03164 2/20 0.47
REV1 Q9UBZ9 1/20 0.47
NPC1 O15118 3/20 0.45
TP53 P04637 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 2/20 0.44
MAPT P10636 1/20 0.44
MGAM O43451 3/20 0.43
GAA P10253 3/20 0.43
SI P14410 3/20 0.43
MGAM2 Q2M2H8 3/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567252 0.85 CYP19A1 (0.53) CYP19A1FAAHMGLLKMT2AREV1
SCHEMBL21051428 0.84 PDE10A (0.51) CYP19A1FAAHMGLLREV1NPC1
SCHEMBL7565376 0.82 FFAR1 (0.55) TP53MAPT
SCHEMBL5372077 0.81 CYP19A1 (0.48) CYP19A1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL5378962 0.80 KMT2A (0.64) CYP19A1KMT2AALDH1A1LMNAGAA
SCHEMBL7564649 0.79 MAOB (0.45) KMT2ANPC1RAB9ASMN1; SMN2MEN1
SCHEMBL7595267 0.78 CNR1 (0.47) CYP19A1FAAHMGLLNPC1RAB9A
SCHEMBL5384888 0.77 HDAC1 (0.55) CYP19A1FAAHMGLLKMT2ANPC1
SCHEMBL5377556 0.77 KMT2A (0.52) KMT2ANPC1RAB9ASMN1; SMN2MEN1
SCHEMBL5377099 0.76 FFAR1 (0.56) ALDH1A1MAPTGAAPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed