SCHEMBL7595267

SCHEMBL7595267

COc1cn(Cc2ccccc2)nc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.47
CNR2 P34972 3/20 0.47
ACHE P22303 2/20 0.47
CYP19A1 P11511 2/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
SLC6A4 P31645 1/20 0.46
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
FAAH O00519 1/20 0.41
MGLL Q99685 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
CHRNA7 P36544 2/20 0.41
ERBB2 P04626 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DAPK1 P53355 1/20 0.41
PDGFRB P09619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567252 0.93 CYP19A1 (0.53) CNR1CNR2CYP19A1FAAHMGLL
SCHEMBL27796924 0.86 SRD5A1 (0.43) CNR1CNR2ACHECYP19A1HTR2A
SCHEMBL11154472 0.79 KMT2A (0.43) CYP19A1HSD17B10
SCHEMBL7567690 0.78 CYP19A1 (0.51) CYP19A1FAAHMGLLMGAMGAA
SCHEMBL7571072 0.77 FFAR1 (0.53) FAAHMGLL
SCHEMBL31200726 0.77 CYP19A1 (0.43) CYP19A1HTR2CERBB2L3MBTL1NPC1
SCHEMBL5393507 0.77 CNR1 (0.50) CNR1CNR2ACHECYP19A1HTR2A
SCHEMBL5376994 0.75 SMN1; SMN2 (0.53) CNR1CNR2ACHECYP19A1HTR2A
SCHEMBL14973897 0.73 P2RX7 (0.43) HSD17B10
SCHEMBL5109055 0.73 CNR1 (0.44) CNR1CNR2ACHECYP19A1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed