SCHEMBL7567252

SCHEMBL7567252

COc1cn(Cc2ccc(OCc3ccccc3)cc2)nc1OCc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.53
FAAH O00519 1/20 0.51
MGLL Q99685 1/20 0.51
REV1 Q9UBZ9 1/20 0.49
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
BCHE P06276 1/20 0.47
NPC1 O15118 3/20 0.47
TP53 P04637 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
PTGS1 P23219 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7595267 0.93 CNR1 (0.47) CYP19A1FAAHMGLLCNR1CNR2
SCHEMBL7567690 0.85 CYP19A1 (0.51) CYP19A1FAAHMGLLREV1BCHE
SCHEMBL7571072 0.83 FFAR1 (0.53) FAAHMGLLTP53
SCHEMBL27796924 0.80 SRD5A1 (0.43) CYP19A1CNR1CNR2NPC1RAB9A
SCHEMBL5385039 0.80 LMNA (0.49) CYP19A1FAAHMGLLCNR1CNR2
SCHEMBL5372207 0.79 SMN1; SMN2 (0.50) CYP19A1FAAHMGLLBCHENPC1
SCHEMBL7569110 0.76 PPARG (0.44) FAAHMGLLNPC1TP53RAB9A
SCHEMBL5372048 0.76 MEN1 (0.51) MEN1ALDH1A1KMT2AL3MBTL1LMNA
SCHEMBL11154472 0.74 KMT2A (0.43) CYP19A1ALDH1A1KMT2A
SCHEMBL6593163 0.74 GAA (0.58) KDM4EMEN1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed