SCHEMBL7567940

SCHEMBL7567940

C=C1CC(c2ccc(SC)cc2)=C1c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.59
PTGS1 P23219 6/20 0.59
GSK3B P49841 1/20 0.39
ALDH1A3 P47895 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GCGR P47871 1/20 0.33
CFTR P13569 1/20 0.33
GOPC Q9HD26 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7566068 0.80 PTGS2 (0.60) PTGS2PTGS1GSK3BKMT2ACFTR
SCHEMBL7567894 0.76 PTGS2 (0.53) PTGS2PTGS1GSK3BALDH1A3MEN1
SCHEMBL7566421 0.74 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL17283465 0.73 PTGS2 (0.63) PTGS2PTGS1GSK3BALDH1A3MEN1
SCHEMBL403028 0.73 PTGS2 (0.63) PTGS2PTGS1GSK3BALDH1A3MEN1
SCHEMBL8654013 0.73 PTGS2 (0.62) PTGS2PTGS1GSK3BALDH1A3MEN1
SCHEMBL5751033 0.72 KMT2A (0.71) PTGS2PTGS1KMT2A
Hydrogen Sulfide SCHEMBL19086306 0.71 PTGS2 (0.61) PTGS2PTGS1GSK3BALDH1A3MEN1
SCHEMBL22477431 0.69 PTGS1 (0.50) PTGS2PTGS1ESR1ESR2KMT2A
SCHEMBL6993410 0.69 PTGS2 (0.56) PTGS2PTGS1GSK3BKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP disclosed
US-5817700-A ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1998-10-06 US disclosed