SCHEMBL7567894

SCHEMBL7567894

CSc1ccc(C2=C(c3ccccc3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.53
PTGS1 P23219 5/20 0.47
ALDH1A3 P47895 1/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
GAA P10253 2/20 0.39
RAB9A P51151 2/20 0.39
GSK3B P49841 1/20 0.39
NPC1 O15118 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
CFTR P13569 1/20 0.37
GOPC Q9HD26 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8654013 0.92 PTGS2 (0.62) PTGS2PTGS1ALDH1A3MEN1KMT2A
SCHEMBL403028 0.84 PTGS2 (0.63) PTGS2PTGS1ALDH1A3MEN1KMT2A
SCHEMBL17283465 0.84 PTGS2 (0.63) PTGS2PTGS1ALDH1A3MEN1KMT2A
Hydrogen Sulfide SCHEMBL19086306 0.81 PTGS2 (0.61) PTGS2PTGS1ALDH1A3MEN1KMT2A
SCHEMBL7212942 0.78 ALDH1A1 (0.53) PTGS2PTGS1KMT2ACYP1A2CYP3A4
SCHEMBL6247727 0.77 PTGS2 (0.57) PTGS2PTGS1ALDH1A3MEN1KMT2A
SCHEMBL7567940 0.76 PTGS2 (0.59) PTGS2PTGS1ALDH1A3MEN1KMT2A
SCHEMBL7566068 0.76 PTGS2 (0.60) PTGS2PTGS1KMT2AGSK3BCFTR
Bicarbonate SCHEMBL29125500 0.76 PTGS2 (0.60) PTGS2ALDH1A3MEN1KMT2ARAB9A
Bicarbonate SCHEMBL28112658 0.76 PTGS2 (0.60) PTGS2ALDH1A3MEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP disclosed
US-5817700-A ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1998-10-06 US disclosed