SCHEMBL7568236

SCHEMBL7568236

Cc1csc(CC(=O)c2ccc(F)c(F)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
NPC1 O15118 4/20 0.36
DPP4 P27487 1/20 0.36
RAB9A P51151 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CHRNA1 P02708 1/20 0.35
CHRNG P07510 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
SLC6A2 P23975 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CHRND Q07001 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778027 0.85 RAB9A (0.43) CES2CES1KMT2AMEN1NPC1
SCHEMBL7832355 0.83 NPC1 (0.47) CES2CES1KMT2AMEN1ALDH1A1
SCHEMBL7850769 0.82 RAB9A (0.55) CES2CES1KMT2AMEN1ALDH1A1
SCHEMBL7833284 0.81 KMT2A (0.48) CES2CES1KMT2AMEN1ALDH1A1
SCHEMBL7832652 0.79 GSK3B (0.44) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL6168851 0.78 RAB9A (0.47) CES2CES1KMT2AMEN1ALDH1A1
SCHEMBL7839557 0.77 NPC1 (0.51) CES2CES1KMT2AMEN1LMNA
SCHEMBL7832513 0.77 CTNNB1 (0.44) CES2CES1KMT2AMEN1ALDH1A1
SCHEMBL7622865 0.77 TDP1 (0.50) KMT2AMEN1ALDH1A1LMNANPC1
SCHEMBL7846518 0.76 CES2 (0.43) CES2CES1KMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP disclosed
US-5817700-A ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1998-10-06 US disclosed