SCHEMBL7569147

SCHEMBL7569147

Cc1cc(NC(C)C)cc2c1OCC2(C)C

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 13/20 0.43
PTGS2 P35354 13/20 0.43
ALOX5 P09917 7/20 0.35
CYP26A1 O43174 1/20 0.31
CYP26B1 Q9NR63 1/20 0.31
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7562111 0.83 PTGS1 (0.42) PTGS1PTGS2ALOX5
SCHEMBL7564292 0.80 PTGS2 (0.43) PTGS1PTGS2ALOX5NOTUM
SCHEMBL7564450 0.80 PTGS2 (0.67) PTGS1PTGS2ALOX5
SCHEMBL672713 0.70 PTGS2 (0.35) PTGS1PTGS2ALOX5NOTUM
SCHEMBL7571234 0.70 PTGS2 (0.35) PTGS1PTGS2ALOX5NOTUM
SCHEMBL17612789 0.68 SSTR5 (0.39) PTGS1PTGS2ALOX5NOTUM
SCHEMBL11404383 0.68 TDP1 (0.46)
SCHEMBL670524 0.67 PTGS2 (0.40) PTGS1PTGS2ALOX5NOTUM
SCHEMBL6154102 0.67 PTGS2 (0.35) PTGS1PTGS2ALOX5NOTUM
SCHEMBL6156608 0.63 PTGS2 (0.32) PTGS1PTGS2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228055-A1 DIHYDROAMINOBENZO[B]- AND [C]FURANS AS RETINOID-LIKE AGENTS Allergan Sales, Inc. (US) 2002-08-07 EP disclosed
WO-2001012618-A1 DIHYDROAMINOBENZO[B]- AND [C]FURANS AS RETINOID-LIKE AGENTS ALLERGAN SALES, INC. (US) 2001-02-22 WO disclosed
US-6093838-A FOR TREATING SKIN-RELATED DISEASES, INCLUDING ACTINIC KERATOSES, ARSENIC KERATOSES, ECZEMA ALLERGAN SALES, INC. (US) 2000-07-25 US disclosed