SCHEMBL7569217

SCHEMBL7569217

O=COc1ccc2[nH]c(-c3ccncc3)nc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
PKN1 Q16512 5/20 0.51
PKN2 Q16513 5/20 0.51
KDM4E B2RXH2 5/20 0.51
HPGD P15428 4/20 0.51
HSD17B10 Q99714 2/20 0.51
RHEB Q15382 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
CBFB Q13951 2/20 0.50
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE3B Q13370 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108052 0.81 ALDH1A1 (0.58) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL6220036 0.80 PKN1 (0.50) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL4248197 0.78 PKN1 (0.55) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL125825 0.77 CBFB (0.81) KDM4EHPGDCBFBNPC1RAB9A
Ridinilazole SCHEMBL413723 0.77 ALDH1A1 (0.66) ALDH1A1PKN1PKN2KDM4EHPGD
Ridinilazole SCHEMBL29379856 0.77 ALDH1A1 (0.66) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL125123 0.76 CBFB (0.63) KDM4EHPGDCYP1A2CYP3A4CYP2C9
SCHEMBL21816537 0.75 CBFB (0.43) ALDH1A1KDM4EHPGDCBFBNPC1
SCHEMBL22772169 0.75 CBFB (0.43) ALDH1A1CYP1A2CYP2C19CBFBMAPT
SCHEMBL10219450 0.75 CBFB (0.43) ALDH1A1KDM4EHPGDHSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194425-A1 SUBSTITUTED BENZIMIDAZOLE Aventis Pharma Deutschland GmbH (DE) 2002-04-10 EP disclosed
WO-2001000610-A1 SUBSTITUTED BENZIMIDAZOLE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-01-04 WO disclosed