Ridinilazole

Ridinilazole

SCHEMBL29379856

c1cc(-c2nc3cc(-c4ccc5[nH]c(-c6ccncc6)nc5c4)ccc3[nH]2)ccn1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.66
KDM4E B2RXH2 4/20 0.66
PKN1 Q16512 4/20 0.66
PKN2 Q16513 4/20 0.66
HPGD P15428 3/20 0.65
RHEB Q15382 2/20 0.65
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
CYP2C9 P11712 1/20 0.65
CYP2C19 P33261 1/20 0.65
HSD17B10 Q99714 1/20 0.65
NPC1 O15118 3/20 0.58
RAB9A P51151 2/20 0.58
GUSB P08236 1/20 0.55
SCD O00767 1/20 0.52
PKM P14618 2/20 0.50
PDE3B Q13370 2/20 0.50
PDE3A Q14432 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ridinilazole SCHEMBL413723 1.00 ALDH1A1 (0.66) ALDH1A1KDM4EPKN1PKN2HPGD
Ridinilazole SCHEMBL17867397 0.93 NPC1 (0.65) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16498509 0.92 KDM4E (0.57) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL6263502 0.91 ALDH1A1 (0.58) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL22906080 0.91 ALDH1A1 (0.58) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL14834116 0.89 KDM4E (0.54) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16499476 0.88 ALDH1A1 (0.65) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16499516 0.88 ALDH1A1 (0.53) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16498482 0.88 ALDH1A1 (0.53) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL19994448 0.87 ALDH1A1 (0.59) ALDH1A1KDM4EPKN1PKN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
US-12318487-B2 Solid tablet dosage form of ridinilazole SUMMIT (OXFORD) LIMITED (GB) 2025-06-03 US claimed
US-20250032515-A1 COMPOSITIONS AND METHODS OF CLOSTRIDIODIDES DIFFICILE TREATMENT, DECOLONIZATION, AND PREVENTION WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2025-01-30 US claimed
US-12115170-B2 Compositions and methods of clostridiodides difficile treatment, decolonization, and prevention WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2024-10-15 US claimed
US-20240277800-A1 PHARMACEUTICAL COMPOSITION COMPRISING MACROCOSINE COMPOUND AND METHOD FOR PREPARING MACROCOSINE COMPOUND A & J SCIENCE CO., LTD. (KR) 2024-08-22 US claimed
US-20240173365-A1 METHODS OF COLONIZING A MICROBIOME, TREATING AND/OR PREVENTING INFLAMMATORY BOWEL DISEASE AND GRAFT VERSUS HOST DISEASE VEDANTA BIOSCIENCES, INC. (US) 2024-05-30 US claimed
EP-4362961-A1 METHODS OF COLONIZING A MICROBIOME, TREATING AND/OR PREVENTING INFLAMMATORY BOWEL DISEASE AND GRAFT VERSUS HOST DISEASE Vedanta Biosciences, Inc. (US) 2024-05-08 EP claimed
WO-2024079245-A1 RIDINILAZOLE FOR TREATING CLOSTRIDIUM DIFFICILE SUMMIT (OXFORD) LIMITED (GB) 2024-04-18 WO claimed
EP-4342484-A1 PHARMACEUTICAL COMPOSITION COMPRISING MACROCOSINE COMPOUND AND METHOD FOR PREPARING MACROCOSINE COMPOUND A&J Science Co.,Ltd. (KR) 2024-03-27 EP claimed
WO-2023278477-A9 METHODS OF COLONIZING A MICROBIOME, TREATING AND/OR PREVENTING INFLAMMATORY BOWEL DISEASE AND GRAFT VERSUS HOST DISEASE VEDANTA BIOSCIENCES, INC. (US) 2023-11-30 WO claimed
WO-2023278477-A1 METHODS OF COLONIZING A MICROBIOME, TREATING AND/OR PREVENTING INFLAMMATORY BOWEL DISEASE AND GRAFT VERSUS HOST DISEASE VEDANTA BIOSCIENCES, INC. (US) 2023-01-05 WO claimed
US-20220378804-A1 COMPOSITIONS AND METHODS OF CLOSTRIDIODIDES DIFFICILE TREATMENT, DECOLONIZATION, AND PREVENTION WISCONSIN ALUMNI RESEARCH FOUNDATION 2022-12-01 US claimed
US-11512068-B2 Process for the preparation of crystalline ridinilazole using acid addition salts SANDOZ AG (CH) 2022-11-29 US claimed
WO-2022245150-A1 PHARMACEUTICAL COMPOSITION COMPRISING MACROCOSINE COMPOUND AND METHOD FOR PREPARING MACROCOSINE COMPOUND 주식회사 에이엔제이사이언스 2022-11-24 WO claimed
US-20220289705-A1 PROCESS FOR THE PREPARATION OF RIDINILAZOLE AND CRYSTALLINE FORMS THEREOF SUMMIT (OXFORD) LIMITED (GB) 2022-09-15 US claimed
US-20220226249-A1 SOLID TABLET DOSAGE FORM OF RIDINILAZOLE SUMMIT (OXFORD) LIMITED (GB) 2022-07-21 US claimed
WO-2022153056-A1 PROCESS FOR PURIFYING RIDINILAZOLE SUMMIT (OXFORD) LIMITED (GB) 2022-07-21 WO claimed
WO-2022153246-A1 SOLID TABLET DOSAGE FORM OF RIDINILAZOLE SUMMIT (OXFORD) LTD. (GB) 2022-07-21 WO claimed
EP-3999502-A1 PROCESS FOR THE PREPARATION OF RIDINILAZOLE AND CRYSTALLINE FORMS THEREOF Summit (Oxford) Limited (GB) 2022-05-25 EP claimed
US-20220143108-A1 METHODS OF DECREASING DYSBIOSIS AND RESTORING A MICROBIOME VEDANTA BIOSCIENCES, INC. (US) 2022-05-12 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA IL1B, IL5, SERPINB1 ALDH1A1 4294/4885KDM4E 4014/4885PKN1 4273/4885
US-11512068-B2 Process for the preparation of crystalline ridinilazole using acid addition salts CYP3A5, CYP3A7, CYP3A4 ALDH1A1 141/4885KDM4E 2756/4885PKN1 2494/4885
US-12318487-B2 Solid tablet dosage form of ridinilazole CYP3A5, CYP3A4, CYP3A7 ALDH1A1 357/4885KDM4E 3535/4885PKN1 1391/4885
US-20220226249-A1 SOLID TABLET DOSAGE FORM OF RIDINILAZOLE CYP3A5, CYP3A4, CYP3A7 ALDH1A1 357/4885KDM4E 3535/4885PKN1 1391/4885
US-20220289705-A1 PROCESS FOR THE PREPARATION OF RIDINILAZOLE AND CRYSTALLINE FORMS THEREOF CYP3A4, CYP3A5, CYP3A7 ALDH1A1 269/4885KDM4E 3581/4885PKN1 1517/4885
US-20240277800-A1 PHARMACEUTICAL COMPOSITION COMPRISING MACROCOSINE COMPOUND AND METHOD FOR PREPARING MACROCOSINE COMPOUND SI, VIP, MLEC ALDH1A1 4777/4885KDM4E 2452/4885PKN1 1819/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.