SCHEMBL7571017

SCHEMBL7571017

N#CC1(NC(=O)C2(CCS(=O)(=O)Cc3ccccc3OC(F)F)CN(C(N)=O)CCO2)CC1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.34
CTSB P07858 5/20 0.34
CTSL P07711 5/20 0.34
CTSK P43235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6062047 0.76 CTSS (0.36) CTSSCTSBCTSLCTSK
SCHEMBL7571020 0.75 CTSS (0.38) CTSSCTSBCTSLCTSK
SCHEMBL6063311 0.72 CTSS (0.49) CTSSCTSBCTSLCTSK
SCHEMBL6063309 0.72 CTSS (0.49) CTSSCTSBCTSLCTSK
SCHEMBL6061996 0.72 CTSS (0.40) CTSSCTSBCTSL
SCHEMBL6739784 0.70 CTSS (0.46) CTSSCTSBCTSLCTSK
SCHEMBL7666715 0.70 CTSS (0.44) CTSSCTSBCTSLCTSK
SCHEMBL7656057 0.70 CTSS (0.40) CTSSCTSBCTSLCTSK
SCHEMBL6063314 0.70 CTSS (0.40) CTSSCTSBCTSLCTSK
SCHEMBL6062055 0.69 CTSS (0.43) CTSSCTSBCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001019808-A1 CHEMICAL COMPOUNDS AND COMPOSITIONS AND THEIR USE AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed