SCHEMBL7656057

SCHEMBL7656057

N#CC1(NC(=O)[C@@H](CNC(=O)N2CCOCC2)S(=O)(=O)Cc2ccccc2OC(F)F)CC1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.40
CTSL P07711 5/20 0.40
CTSB P07858 6/20 0.39
CTSK P43235 3/20 0.39
ADRB1 P08588 2/20 0.39
KMT2A Q03164 1/20 0.36
ADRB2 P07550 1/20 0.35
ADRB3 P13945 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6063314 1.00 CTSS (0.40) CTSSCTSLCTSBCTSKADRB1
SCHEMBL6740847 0.87 ADRB1 (0.41) CTSSCTSLCTSBCTSKADRB1
SCHEMBL7656008 0.84 CTSS (0.47) CTSSCTSLCTSBCTSK
SCHEMBL6063311 0.83 CTSS (0.49) CTSSCTSLCTSBCTSK
SCHEMBL6063309 0.83 CTSS (0.49) CTSSCTSLCTSBCTSK
SCHEMBL6739784 0.81 CTSS (0.46) CTSSCTSLCTSBCTSK
SCHEMBL1557652 0.79 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL1557648 0.79 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL6062346 0.78 CTSS (0.34) CTSSADRB1KMT2AADRB2ADRB3
SCHEMBL7571020 0.76 CTSS (0.38) CTSSCTSLCTSBCTSKKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492362-B1 Compounds and compositions as cathepsin S inhibitors AXYS PHARMACEUTICALS, INC. 2002-12-10 US disclosed