SCHEMBL7571258

SCHEMBL7571258

N=C(N)NC(=O)c1cccc(COc2cccc(-c3cccc(C(=O)NC(=N)N)c3)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 7/20 0.60
MRGPRX4 Q96LA9 2/20 0.60
NPC1 O15118 5/20 0.56
RAB9A P51151 5/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
ALDH1A1 P00352 3/20 0.56
NR1H4 Q96RI1 1/20 0.56
F10 P00742 1/20 0.53
NR4A2 P43354 1/20 0.53
SMPD1 P17405 2/20 0.51
LMNA P02545 2/20 0.51
KDM4E B2RXH2 1/20 0.51
TP53 P04637 1/20 0.51
HTT P42858 1/20 0.51
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454583 0.95 F2 (0.67) F2MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL7579209 0.94 MRGPRX4 (0.59) F2MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL17894403 0.86 SMPD1 (0.69) F2RAB9ANR1H4F10NR4A2
SCHEMBL7569906 0.85 SMPD1 (0.56) F2MRGPRX4NPC1ALDH1A1F10
SCHEMBL7455175 0.83 F2 (0.84) F2MRGPRX4F10
Trifluoroacetic Acid SCHEMBL17894491 0.80 SMPD1 (0.60) F2RAB9ANR1H4F10NR4A2
Hydrochloric Acid SCHEMBL8703334 0.80 KAT6A (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL7452930 0.78 F2 (0.94) F2F10NR4A2
SCHEMBL5175529 0.77 HDAC8 (0.62) ALDH1A1NR1H4
Hydrochloric Acid SCHEMBL8705323 0.76 HDAC8 (0.60) ALDH1A1NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214291-A1 BIPHENYL DERIVATIVES USED AS NHE-3 INHIBITORS MERCK PATENT GmbH (DE) 2002-06-19 EP disclosed
WO-2001021582-A1 BIPHENYL DERIVATIVES USED AS NHE-3 INHIBITORS MERCK PATENT GMBH (DE) 2001-03-29 WO disclosed