SCHEMBL7569906

SCHEMBL7569906

N=C(N)NC(=O)c1ccc(COc2cccc(-c3ccc(C(=O)NC(=N)N)cc3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 3/20 0.56
SPHK2 Q9NRA0 3/20 0.54
F2 P00734 4/20 0.52
MAPT P10636 2/20 0.51
ALDH1A1 P00352 1/20 0.51
MRGPRX4 Q96LA9 2/20 0.50
BCL2L1 Q07817 2/20 0.50
MCL1 Q07820 2/20 0.50
F10 P00742 1/20 0.49
SPHK1 Q9NYA1 1/20 0.49
NPC1 O15118 1/20 0.49
F9 P00740 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7579209 0.92 MRGPRX4 (0.59) SMPD1SPHK2F2MAPTALDH1A1
SCHEMBL7446315 0.87 ITGB3 (0.59) F2MAPTALDH1A1BCL2L1MCL1
SCHEMBL7571258 0.85 F2 (0.60) SMPD1F2ALDH1A1MRGPRX4F10
SCHEMBL7454583 0.83 F2 (0.67) SMPD1F2ALDH1A1MRGPRX4F10
SCHEMBL17894403 0.81 SMPD1 (0.69) SMPD1SPHK2F2F10
SCHEMBL5944125 0.79 SMPD1 (0.79) SMPD1SPHK2MRGPRX4BCL2L1MCL1
SCHEMBL7450042 0.77 F2 (0.83) F2F10
Trifluoroacetic Acid SCHEMBL17894491 0.75 SMPD1 (0.60) SMPD1SPHK2F2F10
SCHEMBL5441715 0.75 RAB9A (0.58) MAPTALDH1A1NPC1
SCHEMBL7448763 0.75 F2 (0.85) F2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214291-A1 BIPHENYL DERIVATIVES USED AS NHE-3 INHIBITORS MERCK PATENT GmbH (DE) 2002-06-19 EP disclosed
WO-2001021582-A1 BIPHENYL DERIVATIVES USED AS NHE-3 INHIBITORS MERCK PATENT GMBH (DE) 2001-03-29 WO disclosed