SCHEMBL7579209

SCHEMBL7579209

N=C(N)NC(=O)c1ccc(-c2cccc(OCc3cccc(C(=O)NC(=N)N)c3)c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 3/20 0.59
F2 P00734 5/20 0.56
NR4A2 P43354 1/20 0.53
ALDH1A1 P00352 4/20 0.53
SMPD1 P17405 3/20 0.53
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
NR1H4 Q96RI1 2/20 0.50
F10 P00742 1/20 0.50
MEN1 O00255 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
SPHK2 Q9NRA0 1/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571258 0.94 F2 (0.60) MRGPRX4F2NR4A2ALDH1A1SMPD1
SCHEMBL7569906 0.92 SMPD1 (0.56) MRGPRX4F2ALDH1A1SMPD1NPC1
SCHEMBL7454583 0.90 F2 (0.67) MRGPRX4F2NR4A2ALDH1A1SMPD1
SCHEMBL17894403 0.83 SMPD1 (0.69) F2NR4A2SMPD1RAB9ANR1H4
SCHEMBL7446315 0.79 ITGB3 (0.59) F2ALDH1A1MAPTHTT
SCHEMBL7455175 0.78 F2 (0.84) MRGPRX4F2F10
Trifluoroacetic Acid SCHEMBL17894491 0.77 SMPD1 (0.60) F2NR4A2SMPD1RAB9ANR1H4
SCHEMBL7450280 0.77 F2 (0.87) F2NR4A2F10
SCHEMBL5944125 0.76 SMPD1 (0.79) MRGPRX4NR4A2SMPD1NR1H4SPHK2
SCHEMBL3565625 0.75 MRGPRX4 (1.00) MRGPRX4NR4A2RAB9ASMN1; SMN2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214291-A1 BIPHENYL DERIVATIVES USED AS NHE-3 INHIBITORS MERCK PATENT GmbH (DE) 2002-06-19 EP disclosed
WO-2001021582-A1 BIPHENYL DERIVATIVES USED AS NHE-3 INHIBITORS MERCK PATENT GMBH (DE) 2001-03-29 WO disclosed