SCHEMBL7572097

SCHEMBL7572097

O=C(O)c1cccc2nc3cccc(Cl)c3nc12

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.69
TSHR P16473 2/20 0.52
HAVCR2 Q8TDQ0 1/20 0.45
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
NQO2 P16083 1/20 0.41
DHODH Q02127 1/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PBRM1 Q86U86 1/20 0.41
PARP1 P09874 1/20 0.40
PIM1 P11309 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
MAPT P10636 3/20 0.40
CYP1A2 P05177 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7568127 0.95 ALDH1A1 (0.71) ALDH1A1TSHRHAVCR2MEN1KMT2A
SCHEMBL5886331 0.85 ALDH1A1 (0.58) ALDH1A1TSHRHAVCR2MEN1KMT2A
SCHEMBL68995 0.83 ALDH1A1 (0.88) ALDH1A1TSHRKMT2AKDM4EHSD17B10
SCHEMBL30548734 0.83 ALDH1A1 (0.88) ALDH1A1TSHRKMT2AKDM4EHSD17B10
SCHEMBL10599968 0.82 ALDH1A1 (0.68) ALDH1A1TSHRMEN1KMT2AKDM4E
Phenazine-1-Carboxylic Acid SCHEMBL29370801 0.82 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AKDM4EHSD17B10
Phenazine-1-Carboxylic Acid SCHEMBL122864 0.82 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AKDM4EHSD17B10
Phenazine-1-Carboxylic Acid SCHEMBL28160016 0.82 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AKDM4EHSD17B10
Phenazine-1-Carboxylic Acid SCHEMBL27884214 0.82 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AKDM4EHSD17B10
SCHEMBL7569010 0.82 ALDH1A1 (0.58) ALDH1A1TSHRHAVCR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9856225-B2 Substituted phenazines as antimicrobial agents UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2018-01-02 US disclosed
US-9856225-B2 Substituted phenazines as antimicrobial agents UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2018-01-02 US disclosed
US-20160355487-A1 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2016-12-08 US disclosed
US-20160355487-A1 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2016-12-08 US disclosed
US-20160355487-A1 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2016-12-08 US disclosed
EP-3086791-A2 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS University of Florida Research Foundation, Inc. (US) 2016-11-02 EP disclosed
WO-2015100331-A2 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-07-02 WO disclosed
WO-2015100331-A2 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-07-02 WO disclosed
EP-0934278-B1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LTD (GB) 2002-09-04 EP disclosed
US-6114332-A BACTERICIDES XENOVA LIMITED (GB) 2000-09-05 US disclosed
EP-0934278-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1999-08-11 EP disclosed
WO-1998017650-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1998-04-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160355487-A1 PHENAZINE DERIVATIVES AS ANTIMICROBIAL AGENTS ROS1, NOX4, NOX5 ALDH1A1 1136/4885TSHR 3298/4885HAVCR2 2506/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.