SCHEMBL7572273

SCHEMBL7572273

CCOc1ccc(Cc2cnc(N)nc2N)c(O)c1-c1ccc(CN2CCOCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.43
USP7 Q93009 1/20 0.41
TLR7 Q9NYK1 1/20 0.40
S1PR1 P21453 1/20 0.40
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557155 0.85 DHFR (0.54) DHFRHTT
SCHEMBL6555136 0.85 DHFR (0.50) DHFR
SCHEMBL6555540 0.81 DHFR (0.49) DHFRHTT
SCHEMBL7572297 0.80 USP7 (0.44) DHFRUSP7
SCHEMBL6555063 0.78 DHFR (0.48) DHFR
SCHEMBL6866050 0.77 DHFR (0.45) DHFR
SCHEMBL6556460 0.77 DHFR (0.54) DHFRHTT
SCHEMBL6555159 0.77 DHFR (0.47) DHFR
SCHEMBL6556639 0.77 DHFR (0.50) DHFR
SCHEMBL6555101 0.76 DHFR (0.52) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230224-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-14 EP disclosed
WO-2001032633-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2001-05-10 WO disclosed