SCHEMBL7572308

SCHEMBL7572308

O=C(O)c1c(NC2CCCCO2)sc2c1CCNC2CN1C(=O)c2cccc(O)c2C1=O

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.35
ALDH1A1 P00352 8/20 0.34
KEAP1 Q14145 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 2/20 0.33
TSHR P16473 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7565443 0.87 PTPN2 (0.38) PTPN1ALDH1A1KEAP1CYP1A2CYP2C9
SCHEMBL7564859 0.86 PARP1 (0.37) PTPN1MEN1KMT2A
SCHEMBL5839246 0.83 PTPN1 (0.46) PTPN1
SCHEMBL5843765 0.80 ALDH1A1 (0.38) ALDH1A1KEAP1CYP1A2CYP2C9CYP2C19
SCHEMBL7155796 0.77 PTPN2 (0.43) PTPN1ALDH1A1KEAP1CYP1A2CYP2C9
SCHEMBL5837672 0.73 PTPN1 (0.50) PTPN1
SCHEMBL7564276 0.72 CYP1A2 (0.39) ALDH1A1CYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL5837045 0.72 PTPN1 (0.52) PTPN1
SCHEMBL7557647 0.72 PTPN1 (0.37) PTPN1ALDH1A1KDM4EMEN1GAA
SCHEMBL5810837 0.71 RAB9A (0.51) PTPN1ALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214060-A2 METHOD OF INHIBITING PROTEIN TYROSINE PHOSPHATASE 1B AND/OR T-CELL PROTEIN TYROSINE PHOSPHATASE AND/OR OTHER PTPASES WITH AN ASP RESIDUE AT POSITION 48 NOVO NORDISK A/S (DK) 2002-06-19 EP disclosed
WO-2001017516-A2 METHOD OF INHIBITING PROTEIN TYROSINE PHOSPHATASE 1B AND/OR T-CELL PROTEIN TYROSINE PHOSPHATASE AND/OR OTHER PTPASES WITH AN ASP RESIDUE AT POSITION 48 NOVO NORDISK A/S (DK) 2001-03-15 WO disclosed