SCHEMBL7572363

SCHEMBL7572363

C#CCN=Cc1cccc(F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.56
RAB9A P51151 7/20 0.56
PKM P14618 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
MAPK1 P28482 1/20 0.56
THPO P40225 1/20 0.56
CHRM5 P08912 1/20 0.56
GRM5 P41594 1/20 0.56
BLM P54132 1/20 0.56
PMP22 Q01453 1/20 0.56
NFE2L2 Q16236 6/20 0.47
MAOB P27338 3/20 0.44
MAOA P21397 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 1/20 0.41
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573586 0.79 NPSR1 (0.45) CYP1A2CYP2D6MAPK1MEN1KMT2A
SCHEMBL7572620 0.79 NPC1 (0.56) NPC1RAB9APKMCYP1A2MAPK1
SCHEMBL7575022 0.79 CHRM5 (0.56) NPC1RAB9ACYP1A2CYP2D6CHRM5
SCHEMBL7573616 0.78 NPC1 (0.41) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL3444467 0.77 LMNA (0.46) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL13107935 0.77 LMNA (0.46) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL3444466 0.77 LMNA (0.46) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9116986 0.76 CA12 (0.33) NPC1CHRM5SMN1; SMN2
SCHEMBL7579153 0.76 CHRM5 (0.60) NPC1RAB9ACYP1A2CYP3A4CHRM5
SCHEMBL2588068 0.74 NPC1 (0.58) NPC1RAB9APKMCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed