Malic Acid

Malic Acid

SCHEMBL7573228

O.O=C(O)CC(O)C(=O)O.[NaH]

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CACNA1CCACNA1DCACNA1FCACNA1SDRD2HTR1BHTR1DHTR1F

The experimentally established mechanism targets of Malic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.88
OR51E2 Q9H255 1/20 0.55
TET2 Q6N021 6/20 0.50
TET3 O43151 2/20 0.50
SLC22A6 Q4U2R8 1/20 0.50
TET1 Q8NFU7 1/20 0.50
KDM4A O75164 2/20 0.48
KDM4C Q9H3R0 2/20 0.48
KDM2A Q9Y2K7 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
GABRR1 P24046 2/20 0.42
LMNA P02545 1/20 0.42
KMO O15229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Malic Acid SCHEMBL4269585 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL7574683 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL13570956 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL10884230 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL10492401 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL7568999 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL17135308 1.00 SMN1; SMN2 (0.88) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL28831630 0.97 SMN1; SMN2 (0.94) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL3408017 0.97 SMN1; SMN2 (0.94) SMN1; SMN2OR51E2TET2TET3SLC22A6
Malic Acid SCHEMBL123090 0.97 SMN1; SMN2 (0.94) SMN1; SMN2OR51E2TET2TET3SLC22A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-52014721-A None JP disclosed
JP-52014720-A None JP disclosed
JP-52014720-A None JP disclosed
JP-52014721-A None JP disclosed
CN-118032449-A Method for rapidly evaluating addition amount of combustion regulator in cigarette paper product on production site 牡丹江恒丰纸业股份有限公司 2024-05-14 CN disclosed
US-20240032579-A1 SALTY TASTE-ENHANCING AGENT TABLEMARK CO., LTD. (JP) 2024-02-01 US disclosed
EP-3442489-B1 SUNSCREEN FORMULATIONS COMPRISING AN OLEOSOME SUSPENSION AND AN ACIDIC BUFFERING SYSTEM BOTANECO INC (CA) 2022-07-06 EP disclosed
US-20190105248-A1 SUNSCREEN FORMULATIONS COMPRISING AN OLEOSOME SUSPENSION AND AN ACIDIC BUFFERING SYSTEM BOTANECO INC. (CA) 2019-04-11 US disclosed
EP-3442489-A1 SUNSCREEN FORMULATIONS COMPRISING AN OLEOSOME SUSPENSION AND AN ACIDIC BUFFERING SYSTEM Botaneco Inc. (CA) 2019-02-20 EP disclosed
WO-2017177334-A1 SUNSCREEN FORMULATIONS COMPRISING AN OLEOSOME SUSPENSION AND AN ACIDIC BUFFERING SYSTEM BOTANECO INC. (CA) 2017-10-19 WO disclosed
US-20140271693-A1 AQUEOUS LIQUID COMPOSITION INTERNATIONAL INSTITUTE OF CANCER IMMUNOLOGY, INC. (JP) 2014-09-18 US disclosed
US-20020045027-A1 Anti-fog resin sheet, anti-fog agent and method article DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-04-18 US disclosed
EP-1184408-A2 Anti-fog resin sheet, anti-fog agent and molded article DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-03-06 EP disclosed
EP-0081236-B1 A COMPOUND SEASONING COMPOSITION, A PROCESS FOR ITS PRODUCTION AND ITS USE AS A FOOD COMPONENT AJINOMOTO CO., INC. (JP) 1986-04-23 EP disclosed
US-4563359-A MIXTURE OF GLUTAMIC ACID WITH SODIUM AND POTASSIUM SALTS AJINOMOTO COMPANY, LIMITED (JP) 1986-01-07 US disclosed
EP-0081236-A1 A compound seasoning composition, a process for its production and its use as a food component AJINOMOTO CO., INC. (JP) 1983-06-15 EP disclosed
JP-S5214721-A PROCESS FOR PREPARATION OF SODIUM MALATE HYDRATE KAWASAKI KASEI CHEM LTD 1977-02-03 JP disclosed
JP-S5214721-A PROCESS FOR PREPARATION OF SODIUM MALATE HYDRATE KAWASAKI KASEI CHEM LTD 1977-02-03 JP disclosed
JP-S5214720-A PROCESS FOR PREPARATION OF SODIUM MALATE HYDRATE KAWASAKI KASEI CHEM LTD 1977-02-03 JP disclosed
JP-S5214720-A PROCESS FOR PREPARATION OF SODIUM MALATE HYDRATE KAWASAKI KASEI CHEM LTD 1977-02-03 JP disclosed