SCHEMBL7573401

SCHEMBL7573401

CS(=O)(=O)OCC#Cc1ccc(Cl)s1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.36
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ADORA3 P0DMS8 1/20 0.30
DRD1 P21728 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571863 0.83 LMNA (0.31) TSHRHTTSMN1; SMN2
SCHEMBL7573562 0.83 KMT2A (0.32) KMT2A
SCHEMBL7581864 0.81
SCHEMBL7575152 0.73 CHRM2 (0.39)
SCHEMBL6200902 0.72 LMNA (0.41) PTGDR2MEN1KMT2A
SCHEMBL7581246 0.69
SCHEMBL4387264 0.69 PTGDR2 (0.39) PTGDR2ADORA3DRD1TSHR
SCHEMBL3452817 0.68 CA12 (0.51) MEN1KMT2AHTT
SCHEMBL31046612 0.68 CYP2D6 (0.44) PTGDR2
SCHEMBL7581858 0.68 CYP2D6 (0.44) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed