SCHEMBL7576271

SCHEMBL7576271

O=C(O)C1CCc2ccccc2C1c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.54
MTNR1A P48039 2/20 0.52
MTNR1B P49286 2/20 0.52
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HIF1A Q16665 1/20 0.51
EDNRA P25101 1/20 0.49
CYP11B2 P19099 1/20 0.47
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
PIN1 Q13526 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C1 Q04828 1/20 0.41
PRCP P42785 1/20 0.41
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12200292 0.87 SIGMAR1 (0.51) SIGMAR1MTNR1AMTNR1BCYP1A2CYP2D6
SCHEMBL27324531 0.83 EDNRA (0.52) SIGMAR1MTNR1AMTNR1BCYP1A2CYP2C19
SCHEMBL8037310 0.79 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A
SCHEMBL901095 0.79 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A
SCHEMBL7901109 0.79 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A
SCHEMBL14226877 0.79 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A
SCHEMBL8055209 0.79 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A
SCHEMBL29568643 0.79 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A
SCHEMBL4931265 0.79 CYP1A2 (0.46) SIGMAR1MTNR1AMTNR1BCYP1A2CYP2D6
SCHEMBL2568184 0.78 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C9CYP2C19HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100769-B1 AMINOMETHYLCARBOXYLIC ACID DERIVATIVES AKZO NOBEL NV (NL) 2002-12-04 EP disclosed
US-6410592-B1 THERAPY FOR CENTRAL NERVOUS SYSTEM DISORDERS, PSYCHOLOGICAL DISORDERS AKZO NOBEL N.V. (NL) 2002-06-25 US disclosed
EP-1100769-A1 AMINOMETHYLCARBOXYLIC ACID DERIVATIVES Akzo Nobel N.V. (NL) 2001-05-23 EP disclosed
WO-2000007978-A1 AMINOMETHYLCARBOXYLIC ACID DERIVATIVES AKZO NOBEL N.V. (NL) 2000-02-17 WO disclosed