L-Norepinephrine

L-Norepinephrine

SCHEMBL7577675

NCC(O)c1ccc(O)c(O)c1.O=C1CC(=O)NC(=O)N1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3

The experimentally established mechanism targets of L-Norepinephrine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 4/20 0.66
ADRB3 known ✓ P13945 4/20 0.66
ADRB1 known ✓ P08588 3/20 0.66
ADRA2A known ✓ P08913 3/20 0.66
ADRA2B known ✓ P18089 3/20 0.66
ADRA2C known ✓ P18825 3/20 0.66
ADRA1D known ✓ P25100 3/20 0.66
ADRA1A known ✓ P35348 2/20 0.66
ADRA1B known ✓ P35368 2/20 0.66
BLM P54132 6/20 0.66
MAPT P10636 5/20 0.66
TDP1 Q9NUW8 5/20 0.66
KDM4E B2RXH2 5/20 0.66
RECQL P46063 4/20 0.66
APEX1 P27695 3/20 0.66
MAPK1 P28482 3/20 0.66
MEN1 O00255 3/20 0.66
KMT2A Q03164 3/20 0.66
TAAR1 Q96RJ0 3/20 0.66
HPGD P15428 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Norepinephrine SCHEMBL7577671 0.84 BLM (0.59) BLMMAPTTDP1KDM4ERECQL
L-Norepinephrine SCHEMBL2610 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
L-Norepinephrine SCHEMBL29460319 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
L-Norepinephrine SCHEMBL3489077 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
Norepinephrine SCHEMBL29399946 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
Norepinephrine SCHEMBL2429869 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
L-Norepinephrine SCHEMBL29371849 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
Norepinephrine SCHEMBL2609 0.81 TDP1 (1.00) BLMMAPTTDP1KDM4ERECQL
L-Norepinephrine SCHEMBL17504429 0.79 TDP1 (0.96) BLMMAPTTDP1KDM4ERECQL
L-Norepinephrine SCHEMBL4155242 0.79 BLM (0.96) BLMMAPTTDP1KDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237913-A2 ANTIGEN PREPARATIONS Cantab Pharmaceuticals Research Limited (GB) 2002-09-11 EP disclosed
US-20010031268-A1 Antigen preparations UNIVERSITY OF NOTTINGHAM (GB) 2001-10-18 US disclosed
WO-2001044278-A2 ANTIGEN PREPARATIONS CANTAB PHARMACEUTICALS RESEARCH LIMITED (GB) 2001-06-21 WO disclosed