SCHEMBL7579129

SCHEMBL7579129

Clc1cccc(C=NCC#Cc2ccc3ccccc3c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.43
MAPT P10636 5/20 0.39
GAA P10253 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GRIN1 Q05586 4/20 0.37
GRIN2B Q13224 4/20 0.37
GRIN2D O15399 2/20 0.37
GRIN3B O60391 2/20 0.37
GRIN2A Q12879 2/20 0.37
GRIN2C Q14957 2/20 0.37
GRIN3A Q8TCU5 2/20 0.37
CYP2A6 P11509 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7579120 1.00 CHRM5 (0.43) CHRM5MAPTGAAKDM4EALDH1A1
SCHEMBL7571168 0.87 KDM4E (0.40) MAPTGAAKDM4EALDH1A1L3MBTL1
SCHEMBL7571171 0.87 KDM4E (0.40) MAPTGAAKDM4EALDH1A1L3MBTL1
SCHEMBL7580460 0.86 L3MBTL1 (0.40) MAPTGAAKDM4EALDH1A1L3MBTL1
SCHEMBL7580453 0.86 L3MBTL1 (0.40) MAPTGAAKDM4EALDH1A1L3MBTL1
SCHEMBL7571671 0.86 CHRM5 (0.50) CHRM5MAPTGAAGRIN1GRIN2B
SCHEMBL7571676 0.86 CHRM5 (0.50) CHRM5MAPTGAAGRIN1GRIN2B
SCHEMBL7578987 0.85 CHRM5 (0.49) CHRM5MAPTGAAKDM4EALDH1A1
SCHEMBL7578981 0.85 CHRM5 (0.49) CHRM5MAPTGAAKDM4EALDH1A1
SCHEMBL7573374 0.82 CHRM5 (0.41) CHRM5MAPTGRIN1GRIN2BGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed