SCHEMBL7581379

SCHEMBL7581379

C#C/C(N)=C\c1ccc(Br)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KMT2A Q03164 4/20 0.40
MAPT P10636 4/20 0.40
LMNA P02545 3/20 0.40
MEN1 O00255 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MAPK1 P28482 2/20 0.40
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40
RECQL P46063 1/20 0.37
SLC22A2 O15244 1/20 0.34
SLC22A1 O15245 1/20 0.34
SLC22A3 O75751 1/20 0.34
PLAU P00749 1/20 0.34
KDM4E B2RXH2 2/20 0.34
RAB9A P51151 1/20 0.34
NOS1 P29475 2/20 0.33
CYP2A6 P11509 1/20 0.33
ALDH1A1 P00352 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7579202 0.79 GRIN2D (0.41) NPC1SMN1; SMN2MAPTLMNASLC22A2
SCHEMBL7575165 0.79 GRIN2D (0.41) SLC22A2SLC22A1SLC22A3PLAUALDH1A1
SCHEMBL7571861 0.79 CAPN1 (0.41) KMT2AMAPTLMNAMEN1NPSR1
SCHEMBL7573612 0.79 MAPT (0.49) KMT2AMAPTLMNAMEN1NPSR1
SCHEMBL7572848 0.78 MCL1 (0.46) SMN1; SMN2KMT2AMAPTLMNAMEN1
SCHEMBL7573585 0.77 HSD17B3 (0.47) KMT2AMAPTMEN1NPSR1ALDH1A1
SCHEMBL7575208 0.75 ALDH1A1 (0.53) SMN1; SMN2KMT2AMAPTLMNAMEN1
SCHEMBL7581521 0.75 ALDH1A1 (0.53) SMN1; SMN2MAPTLMNANPSR1KDM4E
SCHEMBL7571662 0.72 MAPT (0.56) NPC1SMN1; SMN2MAPTMAPK1PLAU
SCHEMBL7575600 0.70 GRIN2D (0.50) SMN1; SMN2LMNAKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed