SCHEMBL7573585

SCHEMBL7573585

C#C/C(N)=C\c1cccc(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.47
ALDH1A1 P00352 2/20 0.46
PKM P14618 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
C1S P09871 1/20 0.39
PARP1 P09874 1/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
HSD11B1 P28845 1/20 0.38
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36
SLC9A1 P19634 1/20 0.36
SLC9A3 P48764 1/20 0.36
SLC9A2 Q9UBY0 1/20 0.36
SLC6A19 Q695T7 1/20 0.36
BACE1 P56817 1/20 0.36
POLB P06746 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572617 0.79 TP53 (0.46) ALDH1A1PKMMEN1KMT2APARP1
SCHEMBL7572362 0.79 MAOB (0.49) PKMPARP1MAPT
SCHEMBL7575017 0.79 GRIN1 (0.47) ALDH1A1PKMMEN1KMT2APARP1
SCHEMBL7581379 0.77 NPC1 (0.41) ALDH1A1MEN1KMT2AMAPTNPSR1
SCHEMBL7572848 0.77 MCL1 (0.46) ALDH1A1MEN1KMT2AAKR1C3MAPT
SCHEMBL27589991 0.76 ALDH1A1 (0.50) HSD17B3ALDH1A1PKMMEN1KMT2A
SCHEMBL7579146 0.75 TAAR1 (0.51) ALDH1A1MEN1KMT2APARP1MAPT
SCHEMBL22202969 0.72 ALDH1A1 (0.56) HSD17B3ALDH1A1PKMMEN1KMT2A
SCHEMBL7573955 0.72 FBP1 (0.57) ALDH1A1MEN1KMT2AMAPT
SCHEMBL15684339 0.71 C1S (0.47) HSD17B3ALDH1A1PKMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed