SCHEMBL758196

SCHEMBL758196

OC(c1cccc(OC(F)(F)C(F)(F)F)c1)c1ccc(F)c(Br)c1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.32
DUT P33316 1/20 0.32
ADAM17 P78536 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950343 0.75 CA1 (0.41) SLC6A4
SCHEMBL3070241 0.73 CETP (0.33)
SCHEMBL13491454 0.70 KDM4E (0.43) SLC6A4DUT
SCHEMBL14033969 0.69 CETP (0.47)
SCHEMBL758195 0.69 EPAS1 (0.31)
SCHEMBL11720083 0.68 MAOB (0.43) SLC6A4
SCHEMBL16233093 0.68 DUT (0.40) SLC6A4DUT
SCHEMBL17064738 0.67 CETP (0.43)
SCHEMBL31067601 0.67 CETP (0.43)
SCHEMBL25237882 0.67 PARP1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954668-B9 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed
EP-1954668-B1 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-09-28 EP disclosed