SCHEMBL7583554

SCHEMBL7583554

COc1ccc(C(C)(C)C(C)=O)cc1C=O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ERN1 O75460 13/20 0.43
TLR2 O60603 1/20 0.42
TLR1 Q15399 1/20 0.42
TLR6 Q9Y2C9 1/20 0.42
LMNA P02545 1/20 0.40
TUBB1 Q9H4B7 1/20 0.40
AOX1 Q06278 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7614307 0.82 ALDH1A1 (0.48) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL9577266 0.82 CYP3A4 (0.48) ALDH1A1TSHRTDP1
SCHEMBL4186655 0.82 ALDH1A1 (0.52) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL31738417 0.82 ALDH1A1 (0.52) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL14242951 0.80 ALDH1A1 (0.50) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL2439167 0.80 CYP19A1 (0.45) ALDH1A1TSHR
SCHEMBL7133759 0.79 ALDH1A1 (0.48) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL7616411 0.79 ALDH1A1 (0.48) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL1186123 0.77 ALDH1A1 (0.50) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL14243153 0.77 ALDH1A1 (0.40) ALDH1A1KDM4ETSHRTDP1ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed